معرفی
Antonio Coluccia is an Associate Professor at the Department of Chemistry and Pharmaceutical Technologies, Sapienza University of Rome. His research integrates computational and experimental approaches to discover novel small molecules with biological activity, focusing on antiviral and anticancer agents.
- PhD in Pharmaceutical Chemistry (2008) from Sapienza University
- Postdoctoral research at Cardiff Welsh School of Pharmacy (funded by Pasteur Institute)
- Subsequent postdoctoral work on anti-tubulin agents at Sapienza University
His research spans structure-based drug design, molecular dynamics, and virtual screening, with a focus on:
- Inhibitors of viral proteins (HIV, SARS-CoV-2, rhinovirus, dengue virus)
- Targeting β-catenin, Grb2, and PDZ domains for cancer therapy
- Development of carbonic anhydrase and lactate dehydrogenase inhibitors
Recent publications highlight advancements in multi-targeting molecules, such as dual-acting compounds against SARS-CoV-2 and anticancer pathways, and novel inhibitors for glioblastoma and chronic myeloid leukemia. His work combines computational modeling (docking, molecular dynamics) with experimental validation (in vitro, in vivo).
Scientific awards include prestigious scholarships from the Pasteur Institute – Fondazione Cenci Bolognetti for international and domestic research. He teaches Laboratory Analysis of Medicines and Medicinal Chemistry courses.
Antonio Coluccia در سایتهای دیگر
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