
About
Giuseppe La Regina is an Associate Professor in Medicinal Chemistry at the Department of Chemistry and Pharmaceutical Technologies, Sapienza University of Rome. His research focuses on designing anti-infective, anti-cancer, and CNS-active agents, with expertise in microwave-assisted synthesis and molecular modeling.
- PhD in Medicinal Chemistry (2005), Sapienza University
- Italian Level 2 Master in Drug Design and Development (2007), University of Pavia
- Graduated in Pharmacy (2001), Sapienza University
His scientific work spans HIV, coronavirus, and tuberculosis drug development, alongside cancer therapies targeting tubulin, beta-catenin, and PDZ domains. He has secured significant grants from Sapienza University and the Italian Ministry of Education.
Recent publications highlight ferroptosis induction in cancer cells, dual-targeting agents for metabolic pathways, and innovative healthcare models. His work integrates computational methods with experimental validation.
- 2018: Publons Peer Review Award
- 2017: National Scientific Qualification for Full Professor
- 2007: Farmindustria Prize for Pharmaceutical Research
He actively supervises PhD students and collaborates on projects related to drug resistance, tumor biology, and viral therapies. His lab facilities are located in Building CU020, Rome.
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